SCHEMBL181391

SCHEMBL181391

CCCC[CH]c1ncc[nH]1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP19A1 P11511 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
TLK2 Q86UE8 3/20 0.33
ALOX5 P09917 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
TXN P10599 1/20 0.32
TXNRD1 Q16881 1/20 0.32
HTR1A P08908 1/20 0.31
TAAR1 Q96RJ0 1/20 0.31
CA1 P00915 1/20 0.30
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL269956 0.88
SCHEMBL3404045 0.81 CYP1A2 (0.38) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL218446 0.81
SCHEMBL27191623 0.75 FAAH (0.38) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL9368459 0.75 FAAH (0.38) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL83280 0.75 FAAH (0.38) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL83282 0.75 FAAH (0.38) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
Bromide SCHEMBL28549910 0.74 FAAH (0.37) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL27233087 0.74 KDM4E (0.37) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9
SCHEMBL3405760 0.73 NPC1 (0.39) CYP1A2CYP3A4CYP2D6CYP19A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112174960-B Toll-like receptor modulating 4, 6-diamino-pyrido [3,2-D ] pyrimidine compounds 吉利德科学公司 2023-10-10 CN disclosed
EP-2401264-A2 PEPTOID OLIGOMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME New York University (US) 2012-01-04 EP disclosed
WO-2010098843-A2 PEPTOID OLIGOMERS, PHARMACEUTICAL COMPOSITIONS AND METHODS OF USING THE SAME NEW YORK UNIVERSITY (US) 2010-09-02 WO disclosed