SCHEMBL1815223

SCHEMBL1815223

Clc1[c]c(Cl)cc(-c2c(Cl)cccc2Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIA1 P42261 2/20 0.40
CACNG8 Q8WXS5 2/20 0.40
SRC P12931 4/20 0.37
CYP2A6 P11509 3/20 0.36
CYP1A2 P05177 3/20 0.36
AHR P35869 1/20 0.36
CNR1 P21554 1/20 0.35
TSHR P16473 2/20 0.35
LMNA P02545 1/20 0.35
CES1 P23141 1/20 0.32
FGFR1 P11362 2/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
RET P07949 1/20 0.31
GRK5 P34947 1/20 0.31
TYRO3 Q06418 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
GRM2 Q14416 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5047790 0.82 GRIA1 (0.40) GRIA1CACNG8SRCCYP2A6CYP1A2
SCHEMBL20072696 0.82 GRIA1 (0.47) GRIA1CACNG8SRCCYP2A6CYP1A2
SCHEMBL15636868 0.77 TTR (0.38) CYP1A2MEN1ALDH1A1KMT2A
SCHEMBL2990875 0.77 SRC (0.41) GRIA1CACNG8SRCCYP2A6CYP1A2
SCHEMBL4448776 0.77 AHR (0.46) GRIA1CACNG8SRCCYP2A6CYP1A2
SCHEMBL8050742 0.77 GRIA1 (0.44) GRIA1CACNG8SRCCYP1A2FGFR1
SCHEMBL3873202 0.76 AHR (0.42) CYP2A6CYP1A2AHRCNR1TSHR
SCHEMBL15635852 0.76 GRIA1 (0.41) GRIA1CACNG8SRCCYP2A6CYP1A2
SCHEMBL4453583 0.75 AHR (0.64) GRIA1CACNG8SRCCYP2A6CYP1A2
SCHEMBL15637371 0.74 CYP2A6 (0.56) CYP2A6TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011063223-A1 TETRAHYDRO-β-CARBOLINE DERIVATIVES, SYNTHESIS AND USE THEREOF SOUTHERN RESEARCH INSTITUTE (US) 2011-05-26 WO disclosed