SCHEMBL18153250

SCHEMBL18153250

c1ccc(C2(c3ncccn3)CNCCO2)nc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.38
ALDH1A1 P00352 3/20 0.32
HPGD P15428 3/20 0.32
HSD17B10 Q99714 3/20 0.32
CYP3A4 P08684 2/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
PLD1 Q13393 1/20 0.32
LDHA P00338 1/20 0.32
LDHB P07195 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 2/20 0.31
OPRM1 P35372 1/20 0.31
MEN1 O00255 1/20 0.31
USP2 O75604 1/20 0.31
CYP2C9 P11712 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL976310 0.87 SLC6A2 (0.37) SLC6A2ALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL15536462 0.81 SLC6A2 (0.36) SLC6A2LDHALDHBCYP1A2CYP2D6
SCHEMBL16053222 0.77 METAP2 (0.33) SLC6A2
SCHEMBL26153825 0.77 SLC6A2 (0.45) SLC6A2ALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL26153822 0.77 SLC6A2 (0.45) SLC6A2ALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL16795106 0.77 SLC6A2 (0.45) SLC6A2ALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL17559201 0.72 SLC6A2 (0.36) SLC6A2ALDH1A1HPGDHSD17B10CYP3A4
SCHEMBL27750340 0.70 GRIN1 (0.44) SLC6A2GRIN1GRIN2AGRIN2BLDHA
SCHEMBL16053646 0.70 DAO (0.35) SLC6A2SLC6A4SLC6A3
SCHEMBL977558 0.70 HTR2A (0.47) SLC6A2OPRM1SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3288939-A1 TRICYCLIC MODULATORS OF TNF SIGNALING AbbVie Inc. (US) 2018-03-07 EP disclosed
WO-2016168641-A1 TRICYCLIC MODULATORS OF TNF SIGNALING ABBVIE INC. (US) 2016-10-20 WO disclosed