SCHEMBL18153251

SCHEMBL18153251

CC(C)c1ncc(-c2ccc3nc4n(c3c2)C(c2ccccc2)COC4)cn1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TNF P01375 8/20 0.37
CCNC P24863 1/20 0.35
CDK8 P49336 1/20 0.35
HDAC6 Q9UBN7 4/20 0.34
HDAC8 Q9BY41 3/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC5 Q9UQL6 1/20 0.34
P2RX7 Q99572 1/20 0.33
TNKS2 Q9H2K2 1/20 0.32
PIK3CA P42336 1/20 0.31
MTOR P42345 1/20 0.31
ATM Q13315 1/20 0.31
ATR Q13535 1/20 0.31
RIPK1 Q13546 1/20 0.31
MAPK1 P28482 1/20 0.31
SCD5 Q86SK9 1/20 0.31
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18150959 0.89 TNF (0.38) TNFCCNCCDK8HDAC6HDAC8
SCHEMBL18151156 0.87 TNF (0.38) TNFCCNCCDK8HDAC6HDAC8
SCHEMBL18150817 0.87 TNF (0.38) TNFCCNCCDK8HDAC6HDAC8
SCHEMBL18150881 0.86 TNF (0.37) TNFCCNCCDK8HDAC6HDAC8
SCHEMBL18150804 0.86 FTO (0.37) TNFCCNCCDK8HDAC6HDAC8
SCHEMBL18150897 0.86 TNF (0.40) TNFCCNCCDK8HDAC6HDAC8
SCHEMBL29795081 0.86 TNF (0.40) TNFCCNCCDK8HDAC6HDAC8
SCHEMBL18151244 0.85 PIK3CA (0.41) TNFCCNCCDK8PIK3CAMTOR
SCHEMBL29795074 0.85 PIK3CA (0.41) TNFCCNCCDK8PIK3CAMTOR
SCHEMBL18153218 0.85 TNF (0.39) TNFCCNCCDK8P2RX7RIPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3288939-A1 TRICYCLIC MODULATORS OF TNF SIGNALING AbbVie Inc. (US) 2018-03-07 EP disclosed
WO-2016168641-A1 TRICYCLIC MODULATORS OF TNF SIGNALING ABBVIE INC. (US) 2016-10-20 WO disclosed