SCHEMBL18153352

SCHEMBL18153352

c1ccc([C@H]2COCc3nc4ccc(-c5cnc(N6CCSCC6)nc5)cc4n32)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TNF P01375 4/20 0.35
AOC3 Q16853 3/20 0.34
EGLN1 Q9GZT9 1/20 0.34
HDAC6 Q9UBN7 5/20 0.32
HDAC8 Q9BY41 4/20 0.32
HDAC1 Q13547 3/20 0.32
HDAC5 Q9UQL6 2/20 0.32
KCNH2 Q12809 1/20 0.32
PTPN11 Q06124 1/20 0.32
MTOR P42345 2/20 0.31
CCNC P24863 1/20 0.31
CDK8 P49336 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31
PIK3CA P42336 1/20 0.30
BRD4 O60885 1/20 0.30
GAK O14976 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18150738 0.91 AOC3 (0.43) TNFAOC3KCNH2MTORPIK3CA
SCHEMBL18150795 0.91 AOC3 (0.43) TNFAOC3KCNH2MTORPIK3CA
SCHEMBL18151375 0.91 AOC3 (0.43) TNFAOC3KCNH2MTORPIK3CA
SCHEMBL31292071 0.89 TNF (0.39) TNFAOC3HDAC6HDAC8HDAC1
SCHEMBL18151071 0.88 AOC3 (0.36) TNFAOC3KCNH2MTORBRD4
SCHEMBL18153272 0.88 AOC3 (0.36) TNFAOC3KCNH2MTORBRD4
SCHEMBL18150982 0.87 TNF (0.34) TNFAOC3HDAC6HDAC8HDAC1
SCHEMBL18150682 0.87 TNF (0.38) TNFAOC3HDAC6HDAC8HDAC1
SCHEMBL18150888 0.87 AOC3 (0.40) TNFAOC3KCNH2MTORPIK3CA
SCHEMBL18153231 0.86 TNF (0.37) TNFAOC3HDAC6HDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3288939-A1 TRICYCLIC MODULATORS OF TNF SIGNALING AbbVie Inc. (US) 2018-03-07 EP claimed
WO-2016168641-A1 TRICYCLIC MODULATORS OF TNF SIGNALING ABBVIE INC. (US) 2016-10-20 WO claimed
EP-3288939-A1 TRICYCLIC MODULATORS OF TNF SIGNALING AbbVie Inc. (US) 2018-03-07 EP disclosed
WO-2016168641-A1 TRICYCLIC MODULATORS OF TNF SIGNALING ABBVIE INC. (US) 2016-10-20 WO disclosed