SCHEMBL18154725

SCHEMBL18154725

Cc1nc(N2CCNCC2)nc(N)c1C1CCNCC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
HPGD P15428 3/20 0.45
KDM4E B2RXH2 2/20 0.45
APAF1 O14727 1/20 0.45
POLB P06746 1/20 0.45
MAPT P10636 1/20 0.45
UBE2N P61088 1/20 0.45
HRH1 P35367 1/20 0.42
USP2 O75604 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
CASP1 P29466 3/20 0.37
CASP4 P49662 1/20 0.37
CASP5 P51878 1/20 0.37
PDE10A Q9Y233 1/20 0.37
HRH4 Q9H3N8 3/20 0.36
HRH3 Q9Y5N1 1/20 0.36
CYP1A2 P05177 2/20 0.36
CYP2C19 P33261 2/20 0.36
CASP7 P55210 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18154724 0.77 GUSB (0.46) ALDH1A1HPGDKDM4EAPAF1POLB
SCHEMBL4476048 0.72 HRH1 (0.43) ALDH1A1HPGDKDM4EAPAF1POLB
SCHEMBL18154763 0.72 SMN1; SMN2 (0.59) ALDH1A1HPGDKDM4EAPAF1POLB
SCHEMBL9488077 0.71 HRH1 (0.59) ALDH1A1HPGDKDM4EAPAF1POLB
Hydrochloric Acid SCHEMBL8582704 0.70 HRH1 (0.57) ALDH1A1HPGDKDM4EAPAF1POLB
SCHEMBL6664557 0.67 HRH1 (0.44) ALDH1A1HPGDKDM4EAPAF1POLB
SCHEMBL1229731 0.67 HRH1 (0.85) ALDH1A1HPGDKDM4EPOLBHRH1
SCHEMBL8962532 0.66 HRH1 (0.61) ALDH1A1HPGDKDM4EAPAF1POLB
SCHEMBL6027662 0.66 HRH1 (0.61) ALDH1A1HPGDKDM4EAPAF1POLB
Hydrochloric Acid SCHEMBL18153315 0.66 HTR2A (0.46) ALDH1A1HPGDKDM4EAPAF1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3283482-A1 PLK4 INHIBITORS Ludwig Institute for Cancer Research Ltd (CH) 2018-02-21 EP disclosed
WO-2016166604-A1 PLK4 INHIBITORS LUDWIG INSTITUTE FOR CANCER RESEARCH LTD (CH) 2016-10-20 WO disclosed