SCHEMBL18159891

SCHEMBL18159891

CNC(=O)c1cccc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(C)c3)cc2)c1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 15/20 0.74
KDR P35968 2/20 0.51
RET P07949 2/20 0.50
CDK8 P49336 2/20 0.50
MEN1 O00255 1/20 0.50
PLK4 O00444 1/20 0.50
CIT O14578 1/20 0.50
AURKA O14965 1/20 0.50
MUSK O15146 1/20 0.50
EPHB6 O15197 1/20 0.50
MAPK13 O15264 1/20 0.50
MLNR O43193 1/20 0.50
MAP3K7 O43318 1/20 0.50
RIPK2 O43353 1/20 0.50
DYRK3 O43781 1/20 0.50
PDE6D O43924 1/20 0.50
NR1I2 O75469 1/20 0.50
STK10 O94804 1/20 0.50
CDK14 O94921 1/20 0.50
ABCB11 O95342 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13529051 0.85 RAF1 (1.00) RAF1KDRRETCDK8MEN1
SCHEMBL13556607 0.84 NPC1 (0.62) RAF1MEN1MAPK13MAPK1MAPK12
SCHEMBL10324287 0.81 RAF1 (0.75) RAF1KDRRETCDK8MEN1
SCHEMBL1506293 0.80 RAF1 (0.67) RAF1KDRRETPLK4AURKA
SCHEMBL15612734 0.80 RAF1 (0.70) RAF1KDRRETMEN1PLK4
SCHEMBL14009183 0.78 RAF1 (0.56) RAF1KDRRETCDK8MEN1
SCHEMBL257694 0.76 MMP13 (0.71) RAF1MEN1KMT2AAR
SCHEMBL14550532 0.76 RAF1 (0.55) RAF1KDRRETCDK8MEN1
SCHEMBL10163566 0.75 RAF1 (0.71) RAF1MEN1BRAFKMT2AAR
SCHEMBL258013 0.75 RAF1 (0.63) RAF1KDRMEN1BRAFKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9994515-B2 Aryl naphthyl methanone oxime(s) and process for preparation thereof COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2018-06-12 US disclosed
US-20160304442-A1 ARYL NAPHTHYL METHANONE OXIME(S) AND PROCESS FOR PREPARATION THEREOF COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2016-10-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160304442-A1 ARYL NAPHTHYL METHANONE OXIME(S) AND PROCESS FOR PREPARATION THEREOF MCL1, CYP11B1, CYP21A2 RAF1 655/4885KDR 4266/4885RET 4633/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.