SCHEMBL18166352

SCHEMBL18166352

CCCc1nnnn1-c1cc(OC(=O)NC(C)c2ccncc2)cc(-c2ccc(C)cc2F)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 2/20 0.40
P2RX2 Q9UBL9 2/20 0.40
PRKACA P17612 2/20 0.36
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
PRKX P51817 2/20 0.36
ROCK1 Q13464 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
RPS6KA5 O75582 1/20 0.36
MAP4K4 O95819 1/20 0.36
PRKCG P05129 1/20 0.36
CDK1 P06493 1/20 0.36
RPS6KB1 P23443 1/20 0.36
CDK2 P24941 1/20 0.36
MAPK1 P28482 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
FLT4 P35916 1/20 0.36
IRAK1 P51617 1/20 0.36
RPS6KA3 P51812 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18166434 0.92 P2RX3 (0.42) P2RX3P2RX2PRKACAGSK3AGSK3B
SCHEMBL18166394 0.88 ROCK1 (0.38) P2RX3P2RX2PRKACAGSK3AGSK3B
SCHEMBL18166308 0.88 P2RX3 (0.55) P2RX3P2RX2
SCHEMBL10245880 0.87 P2RX3 (0.53) P2RX3P2RX2PRKACAGSK3AGSK3B
SCHEMBL18036346 0.87 P2RX3 (0.42) P2RX3P2RX2FAAHPTGS2
SCHEMBL18166431 0.87 P2RX3 (0.43) P2RX3P2RX2MAPK1FAAHPTGS2
SCHEMBL18166293 0.83 P2RX3 (0.57) P2RX3P2RX2PRKACAGSK3AGSK3B
SCHEMBL18166355 0.82 P2RX3 (0.61) P2RX3P2RX2
SCHEMBL18166286 0.81 ROCK1 (0.40) P2RX3P2RX2PRKACAGSK3AGSK3B
SCHEMBL18036317 0.81 P2RX3 (0.42) P2RX3P2RX2FAAHPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2038264-B1 TETRAZOLE-SUBSTITUTED ARYLAMIDES HOFFMANN LA ROCHE (CH) 2016-10-26 EP claimed