SCHEMBL18167147

SCHEMBL18167147

COc1cc(Nc2nc3ccccc3nc2C(N)=O)c(OCC[S+](C)[O-])c(OC)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 5/20 0.39
MAPT P10636 5/20 0.37
THRB P10828 1/20 0.36
SHMT2 P34897 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GAA P10253 1/20 0.36
PKM P14618 1/20 0.36
PIM1 P11309 2/20 0.35
CDC7 O00311 1/20 0.35
PLK4 O00444 1/20 0.35
CHEK1 O14757 1/20 0.35
DCLK1 O15075 1/20 0.35
CHUK O15111 1/20 0.35
PDPK1 O15530 1/20 0.35
DAPK3 O43293 1/20 0.35
DYRK3 O43781 1/20 0.35
JAK2 O60674 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKD3 O94806 1/20 0.35
MAP4K4 O95819 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18167157 0.89 PIK3CG (0.46) PIK3CGMAPTSHMT2KDM4EGAA
SCHEMBL18167163 0.87 PIK3CG (0.44) PIK3CGMAPTBRD4
SCHEMBL18167162 0.86 PIK3CG (0.44) PIK3CGMAPTBRD4
SCHEMBL18167148 0.86 MAPT (0.38) PIK3CGMAPTKDM4EMAPK1PIK3CD
SCHEMBL15192968 0.85 PIK3CG (0.42) PIK3CGMAPTSHMT2KDM4EGAA
SCHEMBL15193666 0.85 MAPT (0.39) PIK3CGMAPTTHRBSHMT2KDM4E
SCHEMBL18167149 0.85 PIK3CG (0.38) PIK3CGMAPTTHRBSHMT2KDM4E
SCHEMBL18167151 0.85 PIK3CG (0.38) PIK3CGMAPTTHRBSHMT2KDM4E
SCHEMBL18167159 0.85 PIK3CG (0.46) PIK3CGMAPT
SCHEMBL15192985 0.85 MAPT (0.46) PIK3CGMAPTTHRBSHMT2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630129-B1 QUINOXALINE DERIVATES MERCK PATENT GMBH (DE) 2016-10-26 EP claimed