SCHEMBL1817074

SCHEMBL1817074

COc1cc2c(O)cc3c(c2cc1N1CCCC(CO)C1)-c1ccccc1C3(C)C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.38
PTPN1 P18031 1/20 0.37
MAPT P10636 1/20 0.36
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
CD274 Q9NZQ7 1/20 0.34
PDE3A Q14432 2/20 0.34
PDE10A Q9Y233 2/20 0.33
HTR1A P08908 1/20 0.33
HTR7 P34969 1/20 0.33
CCR4 P51679 3/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
HPGD P15428 1/20 0.33
MTOR P42345 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
ADRA2B P18089 1/20 0.32
ADRA1A P35348 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8512746 0.93 HTT (0.36) HTTPTPN1MAPTNPC1RAB9A
SCHEMBL1813140 0.85 PTPN1 (0.37) PTPN1MAPTCYP1A2CYP3A4TSHR
SCHEMBL164608 0.80 TSHR (0.41) RAB9AHPGDCYP1A2CYP3A4TSHR
SCHEMBL2021919 0.80 MAPT (0.38) HTTMAPTHTR1ACYP1A2CYP3A4
SCHEMBL8511775 0.78 PDK2 (0.39) HTTPTPN1MAPTHTR7HPGD
SCHEMBL165110 0.76 PDK2 (0.40) PTPN1RAB9AHPGDCYP1A2TSHR
SCHEMBL30125362 0.76 PDK2 (0.40) PTPN1RAB9AHPGDCYP1A2TSHR
SCHEMBL30175150 0.76 MAPT (0.34) HTTPTPN1MAPTNPC1RAB9A
SCHEMBL13988230 0.76 MAPT (0.34) HTTPTPN1MAPTNPC1RAB9A
SCHEMBL1816275 0.75 KDM4E (0.36) PTPN1MAPTHTR1AHPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2494408-B9 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL INC (US) 2015-09-02 EP disclosed
EP-2494408-B1 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL INC (US) 2015-04-15 EP disclosed
EP-2494408-A1 PHOTOCHROMIC MATERIALS Transitions Optical, Inc. (US) 2012-09-05 EP disclosed
WO-2011053615-A1 PHOTOCHROMIC MATERIALS TRANSITIONS OPTICAL, INC. (US) 2011-05-05 WO disclosed