SCHEMBL18171887

SCHEMBL18171887

C[C@H](Nc1cnc2cc(Br)ccc2n1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
NUDT1 P36639 1/20 0.47
MAP4K4 O95819 1/20 0.45
MAPK14 Q16539 3/20 0.43
CCNT1 O60563 1/20 0.42
CDK9 P50750 1/20 0.42
PDGFRB P09619 1/20 0.41
PDGFRA P16234 1/20 0.41
LDHA P00338 1/20 0.41
LDHB P07195 1/20 0.41
EGFR P00533 1/20 0.40
PLK1 P53350 2/20 0.40
MEN1 O00255 1/20 0.40
MAPT P10636 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40
AR P10275 1/20 0.40
PFKFB3 Q16875 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27851794 1.00 NUDT1 (0.47) NUDT1MAP4K4MAPK14CCNT1CDK9
SCHEMBL780421 1.00 NUDT1 (0.47) NUDT1MAP4K4MAPK14CCNT1CDK9
SCHEMBL18171857 0.87 CCNT1 (0.44) MAPK14CCNT1CDK9EGFR
SCHEMBL27868798 0.86 PFKFB3 (0.41) PDGFRBPDGFRAPLK1MEN1MAPT
SCHEMBL27851800 0.86 TNF (0.42) MAPK14EGFRPLK1PFKFB3
SCHEMBL782196 0.86 PFKFB3 (0.41) PDGFRBPDGFRAPLK1MEN1MAPT
SCHEMBL780985 0.86 TNF (0.42) MAPK14EGFRPLK1PFKFB3
SCHEMBL782012 0.84 PFKFB3 (0.47) PDGFRBPDGFRAPLK1PFKFB3
SCHEMBL13049097 0.84 NUDT1 (0.47) NUDT1MAP4K4MAPK14CCNT1CDK9
SCHEMBL780785 0.79 KCNH2 (0.43) CDK9EGFRMEN1MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016170163-A1 SUBSTITUTED QUINOXALINES AND BENZOTRIAZINE P70S6 KINASE INHIBITORS SENTINEL ONCOLOGY LIMITED (GB) 2016-10-27 WO disclosed