SCHEMBL1817195

SCHEMBL1817195

O=C(N1CCc2cc(S(=O)(=O)Cl)ccc21)C(F)(F)F

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.76
CA1 P00915 1/20 0.76
CA2 P00918 1/20 0.76
CA7 P43166 1/20 0.76
CA9 Q16790 1/20 0.76
SMN1; SMN2 Q16637 3/20 0.46
NOTUM Q6P988 3/20 0.46
TSHR P16473 3/20 0.46
HTT P42858 3/20 0.46
LMNA P02545 2/20 0.46
PKM P14618 2/20 0.46
USP2 O75604 1/20 0.46
GAA P10253 1/20 0.46
POLB P06746 1/20 0.44
MAPK1 P28482 1/20 0.44
ADRB2 P07550 2/20 0.43
ADRB1 P08588 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2227782 0.92 CA1 (0.65) CA12CA1CA2CA7CA9
SCHEMBL17858266 0.90 CA12 (0.82) CA12CA1CA2CA7CA9
SCHEMBL7844094 0.86 CA1 (1.00) CA12CA1CA2CA7CA9
SCHEMBL15805654 0.85 CA12 (0.54) CA12CA1CA2CA7CA9
SCHEMBL31513336 0.83 CA12 (0.71) CA12CA1CA2CA7CA9
SCHEMBL29737158 0.82 NOTUM (0.64) SMN1; SMN2NOTUMLMNAPKMMAPK1
SCHEMBL1021359 0.82 NOTUM (0.64) SMN1; SMN2NOTUMLMNAPKMMAPK1
SCHEMBL15805636 0.82 CA1 (0.52) CA12CA1CA2CA7CA9
SCHEMBL2616960 0.81 CA12 (0.60) CA12CA1CA2CA7CA9
SCHEMBL13624158 0.80 NOTUM (0.66) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 38 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025088534-A1 BICYCLIC HETEROCYCLE COMPOUNDS AS TEAD INHIBITOR DONG-A ST CO., LTD. (KR) 2025-05-01 WO disclosed
US-20170158702-A1 MULTIVALENT RAS BINDING COMPOUNDS KYRAS THERAPEUTICS, INC. 2017-06-08 US disclosed
US-20170158702-A1 MULTIVALENT RAS BINDING COMPOUNDS KYRAS THERAPEUTICS, INC. 2017-06-08 US disclosed
WO-2017096045-A1 MULTIVALENT RAS BINDING COMPOUNDS KYRAS THERAPEUTICS, INC. (US) 2017-06-08 WO disclosed
US-20170158702-A1 MULTIVALENT RAS BINDING COMPOUNDS KYRAS THERAPEUTICS, INC. 2017-06-08 US disclosed
WO-2017096045-A1 MULTIVALENT RAS BINDING COMPOUNDS KYRAS THERAPEUTICS, INC. (US) 2017-06-08 WO disclosed
WO-2016097394-A1 BICYCLIC SULFONAMIDE DERIVATIVES AS INVERSE AGONISTS OF RETINOID-RELATED ORPHAN RECEPTOR GAMMA (ROR GAMMA (T)) GALDERMA RESEARCH & DEVELOPMENT (FR) 2016-06-23 WO disclosed
US-9174969-B2 Indoline scaffold SHP-2 inhibitors and cancer treatment method UNIVERSITY OF SOUTH FLORIDA (US) 2015-11-03 US disclosed
US-9174969-B2 Indoline scaffold SHP-2 inhibitors and cancer treatment method UNIVERSITY OF SOUTH FLORIDA (US) 2015-11-03 US disclosed
US-9174969-B2 Indoline scaffold SHP-2 inhibitors and cancer treatment method UNIVERSITY OF SOUTH FLORIDA (US) 2015-11-03 US disclosed
US-7101884-B2 Tyrosine kinase inhibitors MERCK & CO., INC. (US) 2006-09-05 US disclosed
US-20050070546-A1 Tyrosine kinase inhibitors MERCK SHARP & DOHME CORP. 2005-03-31 US disclosed
US-20040220216-A1 Tyrosine kinase inhibitors MERCK SHARP & DOHME CORP. 2004-11-04 US disclosed
WO-2003037252-A2 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-05-08 WO disclosed
WO-2003024969-A1 TYROSINE KINASE INHIBITORS MERCK & CO., INC. (US) 2003-03-27 WO disclosed
EP-1021437-B1 ARYLSULFONYLIMIDAZOLONE DERIVATIVES AS AN ANTITUMOR AGENT DONG WHA PHARM IND CO LTD (KR) 2001-11-14 EP disclosed
EP-1021437-A1 ARYLSULFONYLIMIDAZOLONE DERIVATIVES AS AN ANTITUMOR AGENT DONG WHA PHARMACEUTICAL INDUSTRIAL CO. LTD. (KR) 2000-07-26 EP disclosed
US-5932742-A CHEMICAL INTERMEDIATE TO ACTIVE ANTITUMOR AGENT DONG WHA PHARM. IND. CO., LTD. (KR) 1999-08-03 US disclosed
US-5929103-A ANTICARCINOGENIC AGENTS DONG WHA PHARM. IND. CO., LTD. (KR) 1999-07-27 US disclosed
WO-1998007719-A1 ARYLSULFONYLIMIDAZOLONE DERIVATIVES AS AN ANTITUMOR AGENT DONG WHA PHARM. IND. CO., LTD. (KR) 1998-02-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040220216-A1 Tyrosine kinase inhibitors ERBB2, TYRO3, TIE1 CA12 4613/4885CA1 4738/4885CA2 3420/4885
US-20050070546-A1 Tyrosine kinase inhibitors ERBB2, TYRO3, TIE1 CA12 4613/4885CA1 4738/4885CA2 3420/4885
US-20170158702-A1 MULTIVALENT RAS BINDING COMPOUNDS KRAS, HRAS, NRAS CA12 4020/4885CA1 4444/4885CA2 2873/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.