SCHEMBL7844094

SCHEMBL7844094

NS(=O)(=O)c1ccc2c(c1)CCN2C(=O)C(F)(F)F

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 1.00
CA2 P00918 3/20 1.00
CA9 Q16790 3/20 1.00
CA7 P43166 2/20 1.00
CA12 O43570 1/20 1.00
CA14 Q9ULX7 2/20 0.47
SMN1; SMN2 Q16637 3/20 0.46
LMNA P02545 2/20 0.46
TSHR P16473 2/20 0.46
HTT P42858 2/20 0.46
NOTUM Q6P988 2/20 0.46
USP2 O75604 1/20 0.46
GAA P10253 1/20 0.46
PKM P14618 1/20 0.46
ROCK1 Q13464 1/20 0.45
POLB P06746 1/20 0.44
MAPK1 P28482 1/20 0.44
ADRB2 P07550 2/20 0.43
ADRB1 P08588 2/20 0.43
CYP2C9 P11712 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17858266 0.90 CA12 (0.82) CA1CA2CA9CA7CA12
SCHEMBL1817195 0.86 CA12 (0.76) CA1CA2CA9CA7CA12
SCHEMBL31513336 0.83 CA12 (0.71) CA1CA2CA9CA7CA12
SCHEMBL14058862 0.82 CA12 (0.69) CA1CA2CA9CA7CA12
SCHEMBL2081068 0.80 CA12 (0.67) CA1CA2CA9CA7CA12
SCHEMBL2227782 0.79 CA1 (0.65) CA1CA2CA9CA7CA12
SCHEMBL8801961 0.79 CA1 (0.64) CA1CA2CA9CA7CA12
SCHEMBL14058976 0.78 CA1 (0.64) CA1CA2CA9CA7CA12
SCHEMBL30770403 0.77 ESR1 (0.65) CA1CA2CA9CA7CA12
SCHEMBL20681402 0.77 ESR1 (0.65) CA1CA2CA9CA7CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015142001-A2 COMPOUND HAVING CARDIOTONIC ACTIVITY AND PHARMACEUTICAL COMPOSITION FOR PREVENTING OR TREATING HEART FAILURE, CONTAINING SAME 충남대학교산학협력단 2015-09-24 WO disclosed
EP-1021437-B1 ARYLSULFONYLIMIDAZOLONE DERIVATIVES AS AN ANTITUMOR AGENT DONG WHA PHARM IND CO LTD (KR) 2001-11-14 EP disclosed
EP-1021437-A1 ARYLSULFONYLIMIDAZOLONE DERIVATIVES AS AN ANTITUMOR AGENT DONG WHA PHARMACEUTICAL INDUSTRIAL CO. LTD. (KR) 2000-07-26 EP disclosed
US-5932742-A CHEMICAL INTERMEDIATE TO ACTIVE ANTITUMOR AGENT DONG WHA PHARM. IND. CO., LTD. (KR) 1999-08-03 US disclosed
US-5929103-A ANTICARCINOGENIC AGENTS DONG WHA PHARM. IND. CO., LTD. (KR) 1999-07-27 US disclosed
WO-1998007719-A1 ARYLSULFONYLIMIDAZOLONE DERIVATIVES AS AN ANTITUMOR AGENT DONG WHA PHARM. IND. CO., LTD. (KR) 1998-02-26 WO disclosed