SCHEMBL18172201

SCHEMBL18172201

COCCOc1ccccc1-n1ncc(C(=O)Nc2ccc(C(F)(F)F)cc2F)c1N

nearest known ligand 0.72

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 8/20 0.72
KDM4E B2RXH2 3/20 0.56
HPGD P15428 2/20 0.56
HTT P42858 2/20 0.50
RXFP1 Q9HBX9 1/20 0.49
SCN5A Q14524 1/20 0.49
KMT2A Q03164 1/20 0.47
MALT1 Q9UDY8 1/20 0.45
ALDH1A1 P00352 2/20 0.45
MAPK14 Q16539 4/20 0.43
POLB P06746 1/20 0.43
LCK P06239 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
UGCG Q16739 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18172167 0.93 SCN9A (0.73) SCN9AKDM4EHPGDHTTRXFP1
SCHEMBL18172156 0.79 SCN9A (0.77) SCN9ARXFP1SCN5AKMT2AMAPK14
SCHEMBL18172027 0.77 MAPK14 (0.59) SCN9AHPGDSCN5AKMT2AALDH1A1
SCHEMBL18172103 0.77 SCN9A (0.65) SCN9AKDM4EHPGDSCN5AMALT1
SCHEMBL18172018 0.74 SCN9A (0.72) SCN9ASCN5AMAPK14
SCHEMBL18172235 0.74 SCN9A (0.72) SCN9ASCN5A
SCHEMBL18172225 0.74 SCN9A (0.60) SCN9ASCN5AMALT1MAPK14LCK
SCHEMBL18172073 0.74 HPGD (0.61) SCN9AKDM4EHPGDHTTSCN5A
SCHEMBL18172037 0.73 SCN9A (0.75) SCN9ASCN5AMAPK14
SCHEMBL18172237 0.73 SCN9A (0.72) SCN9ASCN5AMAPK14UGCG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286178-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS Almirall S.A. (ES) 2018-02-28 EP disclosed
WO-2016170009-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS ALMIRALL, S.A. (ES) 2016-10-27 WO disclosed