SCHEMBL18172073

SCHEMBL18172073

CCOC(=O)c1cnn(-c2ccccc2OCCOC)c1N

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.61
ALDH1A1 P00352 3/20 0.61
RAB9A P51151 5/20 0.59
NPC1 O15118 5/20 0.59
TP53 P04637 1/20 0.59
MAPT P10636 8/20 0.54
SMN1; SMN2 Q16637 4/20 0.54
LMNA P02545 1/20 0.54
TSHR P16473 3/20 0.54
HTT P42858 1/20 0.53
MAPK14 Q16539 1/20 0.52
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C19 P33261 1/20 0.51
RECQL P46063 1/20 0.51
HSD17B10 Q99714 1/20 0.51
SCN5A Q14524 1/20 0.48
SCN9A Q15858 1/20 0.48
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17844090 0.88 ALDH1A1 (0.67) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL18497701 0.87 ALDH1A1 (0.63) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL18172027 0.86 MAPK14 (0.59) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL18172002 0.81 ALDH1A1 (0.72) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL17844204 0.81 ALDH1A1 (0.72) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL18172095 0.80 SCN9A (0.60) HPGDALDH1A1MAPTSMN1; SMN2LMNA
SCHEMBL13131101 0.79 ALDH1A1 (0.69) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL31117051 0.79 ALDH1A1 (0.69) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL3520425 0.79 ALDH1A1 (0.69) HPGDALDH1A1RAB9ANPC1TP53
SCHEMBL31116973 0.79 ALDH1A1 (0.69) HPGDALDH1A1RAB9ANPC1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286178-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS Almirall S.A. (ES) 2018-02-28 EP disclosed
WO-2016170009-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS ALMIRALL, S.A. (ES) 2016-10-27 WO disclosed