SCHEMBL18172223

SCHEMBL18172223

Cc1nn(-c2ccccc2Br)c(N)c1C(=O)Nc1ccc(C(F)(F)F)cn1

nearest known ligand 0.81

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 9/20 0.81
SCN5A Q14524 1/20 0.60
WNT3A P56704 4/20 0.51
PTGS1 P23219 3/20 0.48
GAA P10253 1/20 0.46
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
TRPV1 Q8NER1 1/20 0.43
F10 P00742 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18172087 0.89 SCN9A (1.00) SCN9ASCN5AWNT3APTGS1GAA
SCHEMBL18172189 0.89 SCN9A (0.82) SCN9ASCN5AWNT3APTGS1GAA
SCHEMBL18172124 0.89 SCN9A (0.81) SCN9ASCN5AWNT3APTGS1GAA
SCHEMBL18172209 0.88 SCN9A (0.83) SCN9ASCN5AWNT3APTGS1GAA
SCHEMBL18172105 0.87 SCN9A (0.79) SCN9ASCN5APTGS1GAANPC1
SCHEMBL18172061 0.86 SCN9A (0.74) SCN9ASCN5AWNT3APTGS1GAA
SCHEMBL18172227 0.86 SCN9A (0.86) SCN9ASCN5AWNT3APTGS1GAA
SCHEMBL18172232 0.85 SCN9A (0.72) SCN9ASCN5AWNT3ANPC1RAB9A
SCHEMBL18172102 0.84 SCN9A (0.83) SCN9ASCN5AWNT3APTGS1GAA
SCHEMBL18172090 0.84 SCN9A (0.73) SCN9ASCN5APTGS1GAATRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286178-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS Almirall S.A. (ES) 2018-02-28 EP disclosed
WO-2016170009-A1 AMINO-SUBSTITUTED HETEROCYCLIC DERIVATIVES AS SODIUM CHANNEL INHIBITORS ALMIRALL, S.A. (ES) 2016-10-27 WO disclosed