SCHEMBL18172485

SCHEMBL18172485

CC(C)(C)NC(=O)c1cc(-c2ccc(Cl)cc2)cc(-n2nnnc2C2CC2)c1.CC(C)c1nnnn1-c1cc(C(=O)NC(C)(C)C)cc(-c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
P2RY14 Q15391 14/20 0.45
CCR1 P32246 1/20 0.36
OPRD1 P41143 2/20 0.35
SIGMAR1 Q99720 2/20 0.35
PRCP P42785 1/20 0.35
MCHR1 Q99705 3/20 0.35
ADRA2A P08913 1/20 0.34
ADRA2B P18089 1/20 0.34
ADRA2C P18825 1/20 0.34
HSD11B1 P28845 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18172357 0.88 P2RY14 (0.54) P2RY14OPRD1MCHR1
SCHEMBL18172428 0.88 PRCP (0.40) P2RY14PRCPHSD11B1
SCHEMBL18172351 0.86 CNR1 (0.43) P2RY14HSD11B1
SCHEMBL18173388 0.86 P2RX3 (0.44) P2RY14CCR1OPRD1SIGMAR1PRCP
SCHEMBL20533664 0.83 P2RY14 (0.44) P2RY14OPRD1SIGMAR1ADRA2AADRA2B
SCHEMBL20533687 0.83 PRCP (0.42) P2RY14CCR1PRCP
SCHEMBL18184305 0.81 P2RX3 (0.37) P2RY14HSD11B1
SCHEMBL20533797 0.81 P2RY14 (0.47) P2RY14OPRD1SIGMAR1
SCHEMBL20533465 0.81 P2RX3 (0.38) P2RY14CCR1
SCHEMBL18172417 0.81 PRCP (0.38) P2RY14CCR1PRCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286182-A1 TETRAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PSYCHIATRIC DISORDERS F. Hoffmann-La Roche AG (CH) 2018-02-28 EP claimed
WO-2016169902-A1 TETRAZOLE DERIVATIVES FOR USE IN THE TREATMENT OF PSYCHIATRIC DISORDERS F. HOFFMANN-LA ROCHE AG (CH) 2016-10-27 WO claimed