SCHEMBL18173596

SCHEMBL18173596

C=CC(=O)N1CCC[C@H](Cl)C1

nearest known ligand 0.44

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 12/20 0.44
EGFR P00533 5/20 0.44
JAK2 O60674 2/20 0.44
JAK1 P23458 2/20 0.44
BTK Q06187 4/20 0.43
MAP2K7 O14733 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18173568 1.00 JAK3 (0.44) JAK3EGFRJAK2JAK1BTK
SCHEMBL18232327 0.83 JAK3 (0.43) JAK3EGFRJAK2JAK1BTK
SCHEMBL24113542 0.83 JAK3 (0.43) JAK3EGFRJAK2JAK1BTK
SCHEMBL8362428 0.81 CA12 (0.47) JAK3EGFRJAK2JAK1BTK
SCHEMBL16802109 0.81 CA12 (0.47) JAK3EGFRJAK2JAK1BTK
SCHEMBL30208798 0.81 CA12 (0.47) JAK3EGFRJAK2JAK1BTK
SCHEMBL13067829 0.79 JAK3 (0.42) JAK3EGFRJAK2JAK1BTK
SCHEMBL17179528 0.79 JAK3 (0.41) JAK3EGFRJAK2JAK1BTK
SCHEMBL22296413 0.79 JAK3 (0.41) JAK3EGFRJAK2JAK1BTK
SCHEMBL3487800 0.79 ALDH1A1 (0.54) JAK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016170545-A1 PROCESS FOR THE PREPARATION OF 1-[(3R)-3-[4-AMINO-3-(4-PHENOXYPHENVL)-1H- PVRAZOLO[3,4-D]PYRINIIDIN-1-Y1]-1-PIPERIDINVL]-2-PROPEN-1-ONE AND ITS POLYMORPHS THEREOF MSN LABORATORIES PRIVATE LIMITED (IN) 2016-10-27 WO disclosed