SCHEMBL18174472

SCHEMBL18174472

CCc1ccc(-c2ccc3ncc4ccc(=O)n(-c5ccc(N6CCNCC6)c(C(F)(F)F)c5)c4c3n2)cn1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 20/20 0.63
PIK3CA P42336 3/20 0.52
PIK3CD O00329 2/20 0.52
PIK3CG P48736 2/20 0.52
PIK3C3 Q8NEB9 2/20 0.52
RPTOR Q8N122 2/20 0.52
MLST8 Q9BVC4 2/20 0.52
PIK3C2A O00443 1/20 0.52
PIK3C2B O00750 1/20 0.52
PIK3R1 P27986 1/20 0.52
PRKDC P78527 1/20 0.52
CDC42BPA Q5VT25 1/20 0.52
RICTOR Q6R327 1/20 0.52
MAPKAP1 Q9BPZ7 1/20 0.52
PI4KB Q9UBF8 1/20 0.52
CSNK2A2 P19784 1/20 0.50
FECH P22830 1/20 0.50
PIK3CB P42338 1/20 0.50
CLK1 P49759 1/20 0.50
GSK3A P49840 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14239211 0.88 MTOR (0.65) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL15641288 0.88 MTOR (0.69) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL14240434 0.88 MTOR (0.63) MTORPIK3CAPIK3CDPIK3CGPIK3C3
Hydrochloric Acid SCHEMBL18162705 0.88 MTOR (0.65) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL15641404 0.87 MTOR (0.65) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL14240425 0.86 MTOR (0.63) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL15641244 0.86 MTOR (0.78) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL14240421 0.85 MTOR (0.60) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL18174475 0.81 PIK3CA (0.57) MTORPIK3CAPIK3CDPIK3CGPIK3C3
SCHEMBL18174473 0.81 MTOR (0.59) MTORPIK3CAPIK3CDPIK3CGPIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9475812-B2 Pyridonaphthyridine type dual PI3K and mTOR inhibitor and its preparation and use Xuanzhu Pharma Co., Ltd. (CN) 2016-10-25 US disclosed