SCHEMBL18174929

SCHEMBL18174929

COc1cccc2c1NC(=O)C(N)N=C2c1cccc(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NOTCH1 P46531 10/20 0.48
NOTCH3 Q9UM47 7/20 0.48
RBPJ Q06330 3/20 0.44
PTPN5 P54829 1/20 0.42
STK10 O94804 1/20 0.41
SLK Q9H2G2 1/20 0.41
AKR1C3 P42330 1/20 0.41
AKR1C2 P52895 1/20 0.41
GRM5 P41594 1/20 0.40
GRM1 Q13255 1/20 0.40
RORB Q92753 3/20 0.40
PDE4B Q07343 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GAA P10253 1/20 0.39
HPGD P15428 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
RORC P51449 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17030705 0.87 NOTCH1 (0.47) NOTCH1NOTCH3RBPJSTK10SLK
SCHEMBL15631538 0.86 NOTCH1 (0.58) NOTCH1NOTCH3RBPJ
SCHEMBL15622249 0.86 NOTCH1 (0.58) NOTCH1NOTCH3RBPJ
SCHEMBL15608316 0.85 NOTCH1 (0.55) NOTCH1NOTCH3RBPJALDH1A1HPGD
SCHEMBL15622381 0.84 NOTCH1 (0.49) NOTCH1NOTCH3RBPJALDH1A1
SCHEMBL15622403 0.84 NOTCH1 (0.49) NOTCH1NOTCH3RBPJALDH1A1
SCHEMBL15608340 0.84 NOTCH1 (0.56) NOTCH1NOTCH3RBPJSTK10SLK
SCHEMBL17030701 0.83 NOTCH1 (0.46) NOTCH1NOTCH3RBPJ
SCHEMBL15608394 0.82 NOTCH1 (0.61) NOTCH1NOTCH3RBPJSTK10SLK
SCHEMBL15629441 0.82 NOTCH1 (0.61) NOTCH1NOTCH3RBPJSTK10SLK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2897947-B1 ALKYL, FLUOROALKYL-1,4-BENZODIAZEPINONE COMPOUNDS BRISTOL MYERS SQUIBB CO (US) 2016-10-26 EP disclosed