SCHEMBL18175040

SCHEMBL18175040

CC(I)c1ccc(C#N)cn1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.43
KDM4E B2RXH2 4/20 0.43
L3MBTL1 Q9Y468 3/20 0.43
CYP19A1 P11511 1/20 0.38
CYP2A6 P11509 2/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
S1PR3 Q99500 1/20 0.35
HPGD P15428 2/20 0.35
HTT P42858 1/20 0.35
EGLN2 Q96KS0 1/20 0.34
PANK3 Q9H999 4/20 0.34
KCNJ1 P48048 2/20 0.33
AURKA O14965 1/20 0.33
GRK6 P43250 1/20 0.33
KCNH2 Q12809 1/20 0.33
SCN10A Q9Y5Y9 1/20 0.33
GRM5 P41594 1/20 0.33
HPGDS O60760 1/20 0.33
CYP11B1 P15538 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2737290 0.84 ALDH1A1 (0.46) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL19574036 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL22538435 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL20447636 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL20447635 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL15486717 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL29872319 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL22481395 0.81 ALDH1A1 (0.43) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL16311933 0.78 ALDH1A1 (0.41) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6
SCHEMBL8575277 0.76 ALDH1A1 (0.42) ALDH1A1KDM4EL3MBTL1CYP19A1CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2888248-B1 SUBSTITUTED 4-PYRIDONES AND THEIR USE AS INHIBITORS OF NEUTROPHIL ELASTASE ACTIVITY BOEHRINGER INGELHEIM INT (DE) 2016-10-26 EP disclosed