SCHEMBL18184262

SCHEMBL18184262

C=C/C=C(/NC(C)=O)C(=C)OC

nearest known ligand 0.38

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.33
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31
CRBN Q96SW2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL714059 0.82 ALDH1A1 (0.39) ALDH1A1KEAP1NFE2L2HCAR2CRBN
SCHEMBL710767 0.82 ALDH1A1 (0.39) ALDH1A1KEAP1NFE2L2HCAR2CRBN
SCHEMBL18184260 0.78 CRBN (0.31) CRBN
SCHEMBL715075 0.77 CRBN (0.33) ALDH1A1CRBN
SCHEMBL4611736 0.77 CRBN (0.33) ALDH1A1CRBN
SCHEMBL23919967 0.72 ALDH1A1 (0.33) ALDH1A1CRBN
SCHEMBL16168274 0.69
SCHEMBL19937378 0.69
SCHEMBL16543568 0.68
SCHEMBL13896472 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016172631-A2 SUBSTRATE SELECTIVE INHIBITORS OF INSULIN-DEGRADING ENZYME (IDE) AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2016-10-27 WO disclosed