SCHEMBL18189646

SCHEMBL18189646

CCOC(=O)CCCCCOc1ccc(C2=N[C@@](C)(C(=O)O)CS2)c(O)c1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 2/20 0.47
ALDH2 P05091 2/20 0.44
MAOA P21397 1/20 0.44
MAOB P27338 1/20 0.44
BRD4 O60885 1/20 0.43
FFAR1 O14842 1/20 0.43
CNR2 P34972 3/20 0.42
CYSLTR2 Q9NS75 2/20 0.39
CYSLTR1 Q9Y271 2/20 0.39
LTA4H P09960 4/20 0.39
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
PLA2G2A P14555 1/20 0.39
PTPN1 P18031 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18189647 1.00 PDK2 (0.47) PDK2ALDH2MAOAMAOBBRD4
SCHEMBL18189670 0.96 PDK2 (0.47) PDK2ALDH2MAOAMAOBBRD4
SCHEMBL18189671 0.96 PDK2 (0.47) PDK2ALDH2MAOAMAOBBRD4
SCHEMBL18197343 0.93 PDK2 (0.45) PDK2ALDH2MAOAMAOBBRD4
SCHEMBL18189626 0.89 PDK2 (0.44) PDK2ALDH2MAOAMAOBFFAR1
SCHEMBL18189583 0.89 PDK2 (0.44) PDK2ALDH2MAOAMAOBFFAR1
SCHEMBL18197348 0.89 BRD4 (0.47) PDK2ALDH2MAOAMAOBBRD4
SCHEMBL20175897 0.88 PTPN11 (0.45) PDK2CNR2
SCHEMBL20175900 0.88 PTPN11 (0.45) PDK2CNR2
SCHEMBL18189559 0.87 HPGD (0.47) ALDH2CNR2PDE3BPDE3APTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3288557-A1 METABOLICALLY PROGRAMMED METAL CHELATORS AND USES THEREOF University of Florida Research Foundation, Inc. (US) 2018-03-07 EP disclosed
WO-2016176343-A1 METABOLICALLY PROGRAMMED METAL CHELATORS AND USES THEREOF UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INCORPORATED (US) 2016-11-03 WO disclosed