SCHEMBL18190876

SCHEMBL18190876

FC(F)(F)Oc1ccc2[nH]c([AsH2])nc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RUNX1 Q01196 6/20 0.43
CBFB Q13951 3/20 0.43
TRPV1 Q8NER1 2/20 0.43
KIF11 P52732 1/20 0.43
KDM4E B2RXH2 2/20 0.42
CRHBP P24387 1/20 0.42
CRHR2 Q13324 1/20 0.42
GAA P10253 2/20 0.42
KMT2A Q03164 1/20 0.42
SCN10A Q9Y5Y9 1/20 0.41
NPC1 O15118 2/20 0.41
RAB9A P51151 2/20 0.41
GMNN O75496 1/20 0.41
USP2 O75604 1/20 0.41
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18190875 0.87 RUNX1 (0.56) RUNX1CBFBTRPV1KIF11GAA
SCHEMBL1193332 0.81 RUNX1 (0.43) RUNX1CBFBTRPV1KIF11KDM4E
SCHEMBL7066940 0.81 RUNX1 (0.43) RUNX1CBFBTRPV1KIF11KDM4E
SCHEMBL9674984 0.81 NPSR1 (0.53) RUNX1CBFBTRPV1KIF11KDM4E
SCHEMBL2108293 0.81 RUNX1 (0.43) RUNX1CBFBTRPV1KIF11KDM4E
SCHEMBL5683128 0.81 NPC1 (0.48) RUNX1CBFBTRPV1KIF11KDM4E
SCHEMBL11903454 0.81 KDM4E (0.47) RUNX1CBFBTRPV1KIF11KDM4E
SCHEMBL23676457 0.80 SCN10A (0.56) RUNX1CBFBTRPV1KIF11KDM4E
Hydrochloric Acid SCHEMBL9765811 0.79 NPC1 (0.49) RUNX1CBFBTRPV1KIF11KDM4E
SCHEMBL18659785 0.78 TRPV1 (0.50) RUNX1CBFBTRPV1KIF11KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3265448-A1 RILUZOLE PRODRUGS AND THEIR USE Biohaven Pharmaceutical Holding Company Ltd. (US) 2018-01-10 EP disclosed
WO-2016140879-A9 RILUZOLE PRODRUGS AND THEIR USE BIOHAVEN PHARMACEUTICAL HOLDING COMPANY LTD. (US) 2016-11-03 WO disclosed