SCHEMBL18197856

SCHEMBL18197856

Fc1nnc2ccc(-c3cccs3)nn12

nearest known ligand 0.63

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
FYN P06241 6/20 0.56
MET P08581 3/20 0.55
KDM4E B2RXH2 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
PKM P14618 1/20 0.50
RXFP1 Q9HBX9 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11152842 0.83 FYN (0.57) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL2496343 0.77 MET (0.78) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL2495116 0.75 MET (0.80) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL2492967 0.74 MET (0.78) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL18613329 0.72 FYN (1.00) FYN
SCHEMBL2499710 0.72 MET (0.78) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL13888410 0.72 MET (0.78) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL2266182 0.72 MET (1.00) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL2494980 0.72 MET (0.49) FYNMETKDM4ESMN1; SMN2MEN1
SCHEMBL2499862 0.71 FYN (0.46) FYNMETKDM4ESMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966214-B9 TRIAZOLOPYRIDAZINES AS TYROSINE KINASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2017-09-13 EP disclosed
EP-1966214-B1 TRIAZOLOPYRIDAZINES AS TYROSINE KINASE MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2016-11-02 EP disclosed