SCHEMBL18210698

SCHEMBL18210698

C=C(O)CSc1cc(NS(=O)(=O)c2ccc(-c3ccc(OCC)cc3)cc2)c2ccccc2c1O

nearest known ligand 0.79

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.79
POLB P06746 5/20 0.79
KMT2A Q03164 5/20 0.79
TDP2 O95551 4/20 0.79
G6PD P11413 4/20 0.79
CFTR P13569 4/20 0.79
GOPC Q9HD26 4/20 0.79
BLM P54132 4/20 0.79
L3MBTL1 Q9Y468 2/20 0.79
MCL1 Q07820 15/20 0.66
KEAP1 Q14145 8/20 0.66
NFE2L2 Q16236 8/20 0.66
BCL2 P10415 5/20 0.66
BCL2L1 Q07817 5/20 0.66
BCL2A1 Q16548 5/20 0.66
BCL2L2 Q92843 5/20 0.66
SQSTM1 Q13501 2/20 0.66
HKDC1 Q2TB90 5/20 0.65
NSD2 O96028 3/20 0.65
RAB9A P51151 3/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14851464 0.92 MEN1 (0.94) MEN1POLBKMT2ATDP2G6PD
SCHEMBL14851527 0.89 MEN1 (1.00) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210694 0.88 MEN1 (0.62) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210692 0.87 MEN1 (0.68) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210703 0.86 MCL1 (0.83) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210697 0.85 MCL1 (0.77) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210699 0.85 MCL1 (0.83) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210682 0.85 MEN1 (0.65) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210671 0.84 MCL1 (0.82) MEN1POLBKMT2ATDP2G6PD
SCHEMBL18210690 0.84 MEN1 (0.63) MEN1POLBKMT2ATDP2G6PD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9486422-B2 Small molecule inhibitors of Mcl-1 and the uses of thereof THE REGENTS OF THE UNIVERSITY OF MICHIGAN (US) 2016-11-08 US disclosed