SCHEMBL18229059

SCHEMBL18229059

CN(CCCCC(=O)Nc1ccc(C=O)cc1)C(=O)CCN1CCC2(CC1)CC(N(C(=O)O)c1ccccc1-c1ccccc1)C2

nearest known ligand 0.43

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 15/20 0.43
ADRB2 P07550 13/20 0.43
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18229114 0.88 CHRM3 (0.41) CHRM3ADRB2BCHEACHE
SCHEMBL18239050 0.88 CHRM3 (0.43) CHRM3ADRB2
SCHEMBL18238906 0.84 CHRM3 (0.55) CHRM3ADRB2
Trifluoroacetic Acid SCHEMBL18229109 0.77 CHRM3 (0.69) CHRM3ADRB2
Trifluoroacetic Acid SCHEMBL18229089 0.77 CHRM3 (0.56) CHRM3ADRB2
SCHEMBL694787 0.77 CHRM3 (0.63) CHRM3ADRB2
Trifluoroacetic Acid SCHEMBL18229067 0.76 ADRB2 (0.53) CHRM3ADRB2
SCHEMBL18229029 0.75 CHRM3 (0.62) CHRM3ADRB2
SCHEMBL28098391 0.75 CHRM3 (0.56) CHRM3ADRB2
SCHEMBL18229037 0.75 CHRM3 (0.36) CHRM3ADRB2BCHEACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016180348-A1 NITROGEN-CONTAINING SPIRO-HETEROCYCLIC DERIVATIVE HAVING BETA2 RECEPTOR EXCITEMENT AND M RECEPTOR ANTAGONISTIC ACTIVITIES AND APPLICATION THEREOF IN MEDICAMENT 四川海思科制药有限公司 2016-11-17 WO disclosed