SCHEMBL18235652

SCHEMBL18235652

FC(F)(F)c1cc(Oc2ccc(I)cc2)ccc1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AR P10275 4/20 0.49
CHEK2 O96017 2/20 0.43
IDO1 P14902 2/20 0.42
KDR P35968 4/20 0.42
RAF1 P04049 4/20 0.42
BRAF P15056 3/20 0.42
HDAC3 O15379 2/20 0.42
HDAC4 P56524 2/20 0.42
HDAC1 Q13547 2/20 0.42
HDAC7 Q8WUI4 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC10 Q969S8 2/20 0.42
HDAC11 Q96DB2 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42
HDAC9 Q9UKV0 2/20 0.42
HDAC5 Q9UQL6 2/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
CDK8 P49336 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5668761 0.84 PPARG (0.52) ARCHEK2IDO1KDRRAF1
SCHEMBL876272 0.83 AR (0.49) ARCHEK2IDO1KDRRAF1
SCHEMBL6511184 0.83 MAOA (0.50) ARCHEK2IDO1RAF1BRAF
SCHEMBL875870 0.81 AR (0.48) ARCHEK2IDO1KDRRAF1
SCHEMBL2396132 0.81 AR (0.51) ARCHEK2IDO1KDRRAF1
SCHEMBL9106976 0.81 IDO1 (0.49) ARCHEK2IDO1KDRRAF1
SCHEMBL24998721 0.80 PPARG (0.51) ARCHEK2IDO1KDRRAF1
SCHEMBL875873 0.80 AR (0.47) ARCHEK2IDO1KDRRAF1
SCHEMBL13945703 0.80 AR (0.47) ARCHEK2IDO1KDRRAF1
SCHEMBL875588 0.80 IDO1 (0.51) ARCHEK2IDO1KDRRAF1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016180247-A1 BICYCLIC COMPOUND USED AS AN LP-PLA2 INHIBITOR, AND PREPARATION METHOD AND PHARMACEUTICAL USE THEREOF 中国科学院上海药物研究所 2016-11-17 WO disclosed