SCHEMBL1826421

SCHEMBL1826421

C[C@]1(c2ccccc2)CC2(N=C(N)NC2=O)c2cc(Br)ccc2O1

nearest known ligand 0.47

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 14/20 0.47
CTSD P07339 5/20 0.47
HSD11B1 P28845 3/20 0.40
BACE2 Q9Y5Z0 1/20 0.39
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1829335 0.89 BACE1 (0.44) BACE1CTSDHSD11B1
SCHEMBL1827624 0.87 BACE1 (0.53) BACE1CTSDHSD11B1
SCHEMBL1832026 0.87 BACE1 (0.45) BACE1CTSDBACE2
SCHEMBL1823413 0.85 BACE1 (0.45) BACE1CTSD
SCHEMBL1830168 0.85 BACE1 (0.43) BACE1CTSDHSD11B1BACE2OPRM1
SCHEMBL1821336 0.84 BACE1 (0.65) BACE1CTSD
SCHEMBL1828991 0.83 BACE1 (0.42) BACE1CTSDHSD11B1BACE2OPRM1
SCHEMBL1827435 0.82 BACE1 (0.40) BACE1CTSDBACE2OPRM1OPRD1
SCHEMBL1827918 0.81 BACE1 (0.47) BACE1CTSDHSD11B1
SCHEMBL1825825 0.81 CTSD (0.45) BACE1CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2324032-A2 INHIBITORS OF BETA-SECRETASE Vitae Pharmaceuticals, Inc. (US) 2011-05-25 EP disclosed
WO-2010021680-A2 INHIBITORS OF BETA-SECRETASE VITAE PHARMACEUTICALS, INC. (US) 2010-02-25 WO disclosed