SCHEMBL18266201

SCHEMBL18266201

CC(NC(=O)c1ccnc(NC(=O)C2CC2)c1)c1cccc(OCC(F)(F)I)c1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 8/20 0.49
ROCK1 Q13464 6/20 0.49
GSK3B P49841 11/20 0.47
GSK3A P49840 6/20 0.47
BRAF P15056 1/20 0.47
MAPT P10636 5/20 0.47
PRKG1 Q13976 2/20 0.45
CYP2C9 P11712 1/20 0.45
PRKACA P17612 1/20 0.45
PRKACG P22612 1/20 0.45
PRKACB P22694 1/20 0.45
AKT1 P31749 1/20 0.45
ACHE P22303 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2713938 0.93 GSK3B (0.55) ROCK2ROCK1GSK3BGSK3ABRAF
SCHEMBL18266214 0.89 ROCK1 (0.49) ROCK2ROCK1GSK3BGSK3APRKG1
SCHEMBL2714843 0.88 GSK3B (0.54) ROCK2ROCK1GSK3BGSK3ABRAF
SCHEMBL18266794 0.87 ROCK2 (0.47) ROCK2ROCK1GSK3BGSK3ABRAF
SCHEMBL2717508 0.86 ROCK2 (0.49) ROCK2ROCK1GSK3BGSK3ABRAF
SCHEMBL2715734 0.86 ROCK2 (0.49) ROCK2ROCK1GSK3BGSK3ABRAF
SCHEMBL15351218 0.86 GSK3B (0.51) ROCK2ROCK1GSK3BGSK3ABRAF
SCHEMBL2715733 0.86 ROCK2 (0.49) ROCK2ROCK1GSK3BGSK3ABRAF
SCHEMBL18266117 0.84 ACACB (0.51) GSK3BGSK3AMAPT
SCHEMBL2715498 0.83 GSK3B (0.58) GSK3BGSK3AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed