SCHEMBL18266341

SCHEMBL18266341

Cc1cc(C(=O)NCc2cccc(OC(C)(F)F)c2F)cc(NC(=O)C(C)C)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.47
RIPK1 Q13546 3/20 0.42
ADORA2A P29274 1/20 0.41
ADORA2B P29275 1/20 0.41
ADORA1 P30542 1/20 0.41
CHRM4 P08173 1/20 0.40
KCNB1 Q14721 1/20 0.38
MAPT P10636 3/20 0.37
GSK3B P49841 2/20 0.37
EPHX2 P34913 3/20 0.37
ALDH1A1 P00352 2/20 0.37
RAB9A P51151 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
ALOX5 P09917 1/20 0.37
PPARG P37231 2/20 0.36
HSD17B13 Q7Z5P4 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2714691 0.94 RIPK1 (0.48) SCN9ARIPK1ADORA2AADORA2BADORA1
SCHEMBL18266494 0.89 RIPK1 (0.42) SCN9ARIPK1ADORA2AADORA2BADORA1
SCHEMBL18266542 0.89 RIPK1 (0.42) SCN9ARIPK1ADORA2AADORA2BADORA1
SCHEMBL2714773 0.85 SCN9A (0.50) SCN9ACHRM4EPHX2ALDH1A1MEN1
SCHEMBL2715976 0.84 RIPK1 (0.57) RIPK1ADORA2AADORA2BADORA1EPHX2
SCHEMBL18266303 0.84 SCN9A (0.47) SCN9ARIPK1CHRM4KCNB1MAPT
SCHEMBL2715536 0.84 RIPK1 (0.48) SCN9ARIPK1ADORA2AADORA2BADORA1
SCHEMBL18266538 0.83 KCNB1 (0.50) SCN9ARIPK1KCNB1GSK3BPPARG
SCHEMBL2714267 0.83 RIPK1 (0.48) RIPK1ADORA2AADORA2BADORA1EPHX2
SCHEMBL18266345 0.83 SCN9A (0.48) SCN9ARIPK1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2630122-B1 ARYLAMIDE DERIVATIVES AS TTX-S BLOCKERS RAQUALIA PHARMA INC (JP) 2016-11-30 EP disclosed