SCHEMBL1828811

SCHEMBL1828811

[CH2]C(O)N=C(C)C

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10949634 0.67
SCHEMBL6444106 0.65
SCHEMBL5663048 0.65
SCHEMBL3336286 0.62
SCHEMBL12712177 0.62 ALDH1A1 (0.31)
SCHEMBL18621322 0.57
SCHEMBL15676 0.57
SCHEMBL212534 0.57
SCHEMBL210425 0.57
SCHEMBL8675003 0.56

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116634870-A Herbicidal combinations 安道麦阿甘有限公司 2023-08-22 CN claimed
CN-116634870-A Herbicidal combinations 安道麦阿甘有限公司 2023-08-22 CN disclosed
US-20230247987-A1 THE USE OF SAFENERS TO IMPROVE TOLERANCE OF ACCASE TOLERANT SORGHUM CROP TO HERBICIDES ADAMA AGAN LTD. (IL) 2023-08-10 US disclosed
WO-2023131947-A1 PROCESS FOR THE PREPARATION OF ARYLOXYPHENOXYPROPIONIC ACID DERIVATIVES IN A NON POLAR SOLVENT WITH A TERTIARY AMINE CATALYST ADAMA AGAN LTD. (IL) 2023-07-13 WO disclosed
EP-4209486-A1 PROCESS FOR THE PREPARATION OF ARYLOXYPHENOXYPROPIONIC ACID DERIVATIVES IN A NON POLAR SOLVENT WITH A TERTIARY AMINE CATALYST Adama Agan Ltd. (IL) 2023-07-12 EP disclosed
WO-2021260681-A1 THE USE OF SAFENERS TO IMPROVE TOLERANCE OF ACCASE TOLERANT SORGHUM CROP TO HERBICIDES ADAMA AGAN LTD. (IL) 2021-12-30 WO disclosed
US-20210022342-A1 THE USE OF SAFENERS TO IMPROVE RESISTANCE OF RICE CROP TO HERBICIDES ADAMA AGAN LTD. (IL) 2021-01-28 US disclosed
EP-3768086-A1 THE USE OF SAFENERS TO IMPROVE RESISTANCE OF RICE CROP TO HERBICIDES Adama Agan Ltd. (IL) 2021-01-27 EP disclosed
WO-2019183180-A1 THE USE OF SAFENERS TO IMPROVE RESISTANCE OF RICE CROP TO HERBICIDES ADAMA AGAN LTD. (IL) 2019-09-26 WO disclosed
EP-1555876-B2 COMBINATIONS OF ARYLOXYPHENOXYPROPIONATES AND SAFENERS AND THEIR USE FOR INCREASING WEED CONTROL BAYER CROPSCIENCE AG (DE) 2011-05-11 EP disclosed
EP-1728430-A1 Herbicidal agents Bayer CropScience GmbH (DE) 2006-12-06 EP disclosed
US-20060014643-A1 Combinations of aryloxyphenoxypropionates and safeners and their use for increasing weed control BAYER CROPSCIENCE GMBH (DE) 2006-01-19 US disclosed
WO-2005092105-A1 HERBICIDE COMBINATION BAYER CROPSCIENCE GMBH (DE) 2005-10-06 WO disclosed
EP-1555876-A2 COMBINATIONS OF ARYLOXYPHENOXYPROPIONATES AND SAFENERS AND THEIR USE FOR INCREASING WEED CONTROL Bayer CropScience GmbH (DE) 2005-07-27 EP disclosed
WO-2004034788-A2 COMBINATIONS OF ARYLOXYPHENOXYPROPIONATES AND SAFENERS AND THEIR USE FOR INCREASING WEED CONTROL BAYER CROPSCIENCE GMBH (DE) 2004-04-29 WO disclosed
EP-1104239-A1 HERBICIDES WITH ACYLATED AMINOPHENYLSULFONYL UREA Aventis CropScience GmbH (DE) 2001-06-06 EP disclosed
EP-1053679-A1 Herbicidal compositions AVENTIS CROPSCIENCE S.A. (FR) 2000-11-22 EP disclosed
WO-2000008932-A1 HERBICIDES WITH ACYLATED AMINOPHENYLSULFONYL UREA AVENTIS CROPSCIENCE GMBH (DE) 2000-02-24 WO disclosed
US-5401700-A Plant protection agents based on pyrazolecarboxylic acid derivatives HOECHST AKTIENGESELLSCHAFT (DE) 1995-03-28 US disclosed
EP-0276741-A2 Process for the preparation of propionic-acid derivatives CIBA-GEIGY AG (CH) 1988-08-03 EP disclosed