SCHEMBL18288796

SCHEMBL18288796

Cc1nc2c(F)cc(-c3nc(N)ncc3F)cc2n1CC1CC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 19/20 0.56
CDK6 Q00534 15/20 0.56
CDK2 P24941 4/20 0.56
CDK1 P06493 6/20 0.54
CCNB1 P14635 4/20 0.54
CCNE1 P24864 4/20 0.54
CCND3 P30281 12/20 0.51
CDK7 P50613 2/20 0.51
CDK9 P50750 2/20 0.51
CCNA2 P20248 1/20 0.51
CCND1 P24385 11/20 0.46
GRIN2B Q13224 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18288783 0.82 CDK4 (0.52) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL18288744 0.79 CDK4 (0.55) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL18288760 0.79 CDK4 (0.55) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL18288902 0.78 CDK4 (0.56) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL29402856 0.76 CDK4 (0.55) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL16892106 0.76 CDK4 (0.55) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL30818384 0.76 CDK4 (0.55) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL18288742 0.75 CDK4 (0.45) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL18288992 0.75 CDK4 (0.56) CDK4CDK6CDK2CDK1CCNB1
SCHEMBL18288912 0.75 CDK4 (0.53) CDK4CDK6CDK2CDK1CCNB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016192630-A1 COMPOUND HAVING KINASE INHIBITING ACTIVITY, METHOD OF PREPARING SAME, AND USE OF SAME 中国科学院上海药物研究所 2016-12-08 WO disclosed