SCHEMBL18288902

SCHEMBL18288902

Cc1nc2c(F)cc(-c3nc(N)ncc3F)cc2n1C1CCCCC1

nearest known ligand 0.56

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 20/20 0.56
CDK6 Q00534 17/20 0.56
CDK2 P24941 15/20 0.56
CCNE1 P24864 3/20 0.53
CDK1 P06493 6/20 0.52
CCNB1 P14635 2/20 0.52
CCND3 P30281 4/20 0.50
CCNA2 P20248 2/20 0.50
CDK7 P50613 4/20 0.49
CDK9 P50750 4/20 0.49
CDK5 Q00535 1/20 0.49
CCND1 P24385 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18288744 0.99 CDK4 (0.55) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL18288760 0.97 CDK4 (0.55) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL18288742 0.86 CDK4 (0.45) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL19089070 0.86 CDK4 (0.55) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL18288992 0.85 CDK4 (0.56) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL15252502 0.81 CDK4 (0.54) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL31066374 0.81 CDK4 (0.54) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL18288796 0.78 CDK4 (0.56) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL18823109 0.77 CDK4 (0.56) CDK4CDK6CDK2CCNE1CDK1
SCHEMBL4246503 0.77 ALDH1A1 (0.38) CDK4CDK6CDK2CCNE1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016192630-A1 COMPOUND HAVING KINASE INHIBITING ACTIVITY, METHOD OF PREPARING SAME, AND USE OF SAME 中国科学院上海药物研究所 2016-12-08 WO disclosed