SCHEMBL18293530

SCHEMBL18293530

CCCC(C#N)(CCC)c1ccccn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KCNH2 Q12809 2/20 0.35
SLC22A2 O15244 1/20 0.35
SLC22A1 O15245 1/20 0.35
PGR P06401 1/20 0.35
THRB P10828 1/20 0.35
ADRB3 P13945 1/20 0.35
OPRK1 P41145 1/20 0.35
BLM P54132 1/20 0.35
PMP22 Q01453 1/20 0.35
PDE3A Q14432 1/20 0.35
SLC47A1 Q96FL8 1/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GAA P10253 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246245 0.86 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1KCNH2SLC22A2SLC22A1
SCHEMBL10449753 0.83 SMN1; SMN2 (0.41) SMN1; SMN2L3MBTL1KCNH2SLC22A2SLC22A1
SCHEMBL11537649 0.79 KCNH2 (0.55) SMN1; SMN2L3MBTL1KCNH2SLC22A2SLC22A1
SCHEMBL6888537 0.76 CHRM2 (0.36) SMN1; SMN2L3MBTL1KCNH2SLC22A2SLC22A1
SCHEMBL15693459 0.75 SMN1; SMN2 (0.44) SMN1; SMN2L3MBTL1KCNH2SLC22A2SLC22A1
SCHEMBL21191856 0.74 SMN1; SMN2 (0.47) SMN1; SMN2L3MBTL1KCNH2SLC22A2SLC22A1
SCHEMBL18427298 0.74 SMN1; SMN2 (0.47) SMN1; SMN2L3MBTL1KCNH2SLC22A2SLC22A1
SCHEMBL14434214 0.73
SCHEMBL6996539 0.73 SMN1; SMN2 (0.48) SMN1; SMN2L3MBTL1TDP1GAAMEN1
SCHEMBL13342069 0.73 SMN1; SMN2 (0.54) SMN1; SMN2L3MBTL1BLMALOX15TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1729772-B1 HETEROARYL PIPERIDINE GLYCINE TRANSPORTER INHIBITORS MERCK SHARP & DOHME (US) 2016-12-07 EP disclosed