SCHEMBL11537649

SCHEMBL11537649

CC(C)N(CCC(C#N)(CCN(C(C)C)C(C)C)c1ccccn1)C(C)C

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.55
BLM P54132 2/20 0.55
CYP3A4 P08684 2/20 0.55
TSHR P16473 2/20 0.55
SLC22A2 O15244 1/20 0.55
SLC22A1 O15245 1/20 0.55
PGR P06401 1/20 0.55
THRB P10828 1/20 0.55
ADRB3 P13945 1/20 0.55
OPRK1 P41145 1/20 0.55
PMP22 Q01453 1/20 0.55
PDE3A Q14432 1/20 0.55
SLC47A1 Q96FL8 1/20 0.55
ALOX15 P16050 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
CHRM2 P08172 3/20 0.36
CHRM4 P08173 2/20 0.36
CHRM5 P08912 2/20 0.36
CHRM1 P11229 2/20 0.36
CHRM3 P20309 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11238412 0.92 SLC22A2 (0.51) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL11236930 0.89 SLC22A2 (0.51) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL11536797 0.86 KCNH2 (0.44) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL10638784 0.85 BLM (0.55) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL10956631 0.82 SLC22A2 (0.43) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL10952757 0.81 SLC22A2 (0.40) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL9581143 0.81 CYP3A4 (0.60) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL10633053 0.81 SLC22A2 (0.48) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL10516737 0.80 CYP3A4 (0.50) KCNH2BLMCYP3A4TSHRSLC22A2
SCHEMBL18293530 0.79 SMN1; SMN2 (0.41) KCNH2BLMCYP3A4TSHRSLC22A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4153797-A α-Aryl-α, α-bis[ω- (disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1979-05-08 US disclosed
US-4107205-A α-Aryl-α,α-bis[ω-(disubstituted amino)alkyl]acetamides and related compounds G. D. SEARLE & CO. (US) 1978-08-15 US disclosed