SCHEMBL1829683

SCHEMBL1829683

CCC(C(=O)O)n1ccc(-c2ccc(OC)cc2)c1-c1ccc(C#N)cc1C

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 1/20 0.44
HRH1 P35367 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
MAPK1 P28482 1/20 0.41
HSD17B10 Q99714 1/20 0.41
MAPK14 Q16539 1/20 0.38
THRB P10828 1/20 0.37
GRM2 Q14416 1/20 0.37
XDH P47989 1/20 0.37
PTPN11 Q06124 1/20 0.36
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
APP P05067 1/20 0.36
CYP2C19 P33261 1/20 0.36
EGLN1 Q9GZT9 2/20 0.36
RXFP1 Q9HBX9 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1829774 0.85 HRH2 (0.41) HRH2HRH1KDM4EMAPK14GRM2
SCHEMBL1829684 0.78 HRH2 (0.45) HRH2HRH1HSD17B10MAPK14GRM2
SCHEMBL1828357 0.74 GRM2 (0.42) HRH2HRH1MAPK14GRM2FNTA
SCHEMBL7229011 0.74 HRH2 (0.47) HRH2HRH1KDM4EALDH1A1HPGD
SCHEMBL1829979 0.72 HRH2 (0.40) HRH2HRH1MAPK14GRM2EGLN1
SCHEMBL2029562 0.69 PTGS1 (0.46) HRH2HRH1KDM4EALDH1A1HPGD
SCHEMBL247807 0.69 PLAU (0.42) SMN1; SMN2APPCYP2C19
SCHEMBL1828903 0.69 GRM2 (0.38) HRH2HRH1MAPK14GRM2FNTA
SCHEMBL247116 0.68 PLAU (0.38) SMN1; SMN2ALDH1A1APPCYP2C19
SCHEMBL1828937 0.67 HRH2 (0.40) HRH2HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2315590-A1 PYRROLE INHIBITORS OF S-NITROSOGLUTATHIONE REDUCTASE N30 Pharmaceuticals, LLC (US) 2011-05-04 EP disclosed
WO-2010019909-A1 PYRROLE INHIBITORS OF S-NITROSOGLUTATHIONE REDUCTASE N30 PHARMACEUTICALS, LLC (US) 2010-02-18 WO disclosed