SCHEMBL1830188

SCHEMBL1830188

COc1ccc2nc(C(=O)N3CCC4(CC3)CC(=O)c3cc(N5CCS(O)(O)CC5)ccc3O4)cc(OC)c2c1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
ACACB O00763 6/20 0.40
CYP19A1 P11511 1/20 0.40
KDM4E B2RXH2 4/20 0.40
ALDH1A1 P00352 4/20 0.40
GAA P10253 4/20 0.40
HPGD P15428 2/20 0.40
CASP1 P29466 2/20 0.40
HSD17B10 Q99714 2/20 0.40
KMT2A Q03164 2/20 0.40
GLA P06280 2/20 0.40
CYP1A2 P05177 1/20 0.40
CASP7 P55210 1/20 0.40
ACACA Q13085 3/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1832467 0.90 ALDH1A1 (0.47) CA1CA2CA7CA9ACACB
SCHEMBL1830674 0.88 CA1 (0.43) CA1CA2CA7CA9ACACB
SCHEMBL1830410 0.86 ACACB (0.42) CA1CA2CA7CA9ACACB
SCHEMBL1828716 0.86 HDAC3 (0.49) ACACBCYP19A1KDM4EALDH1A1GAA
SCHEMBL1813933 0.86 ACACB (0.45) ACACBACACAHDAC3HDAC4HDAC1
SCHEMBL1828229 0.85 CYP19A1 (0.46) CA1CA2CA7CA9ACACB
SCHEMBL1829262 0.85 CA1 (0.44) CA1CA2CA7CA9ACACB
SCHEMBL1832752 0.84 ACACB (0.50) ACACBCYP19A1ACACA
SCHEMBL1831980 0.83 HTR2A (0.44) CA1CA2CA7CA9ACACB
SCHEMBL1830323 0.82 ALDH1A1 (0.42) CA1CA2CA7CA9ACACB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1910375-B1 SPIROCHROMANONE DERIVATIVES AS ACETYL COENZYME A CARBOXYLASE (ACC) INHIBITORS MERCK SHARP & DOHME (US) 2011-05-11 EP claimed