SCHEMBL1830898

SCHEMBL1830898

O=c1cc(-c2ccncn2)nc2n1CCCCC2C(F)Cc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.43
CYP2D6 P10635 5/20 0.43
CYP1A2 P05177 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1832035 0.89 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL1834769 0.83 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL1833225 0.82 GSK3B (0.46) GSK3BCYP2D6CYP1A2
SCHEMBL1835397 0.81 GSK3B (0.44) GSK3BCYP2D6CYP1A2
SCHEMBL1828778 0.79 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL1830440 0.79 GSK3B (0.47) GSK3BCYP2D6
SCHEMBL1834667 0.77 GSK3B (0.51) GSK3BCYP2D6CYP1A2
SCHEMBL2065123 0.76 GSK3B (0.47) GSK3BCYP2D6
SCHEMBL1832336 0.76 GSK3B (0.47) GSK3BCYP2D6
SCHEMBL1836064 0.76 GSK3B (0.45) GSK3BCYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2011525908-A 2011-09-29 JP claimed
EP-2321315-A2 SUBSTITUTED ALKYL PYRIMIDIN-4-ONE DERIVATIVES Mitsubishi Tanabe Pharma Corporation (JP) 2011-05-18 EP claimed
WO-2009156864-A2 SUBSTITUTED ALKYL PYRIMIDIN-4-ONE DERIVATIVES MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-12-30 WO claimed
EP-2321315-A2 SUBSTITUTED ALKYL PYRIMIDIN-4-ONE DERIVATIVES Mitsubishi Tanabe Pharma Corporation (JP) 2011-05-18 EP disclosed
WO-2009156864-A2 SUBSTITUTED ALKYL PYRIMIDIN-4-ONE DERIVATIVES MITSUBISHI TANABE PHARMA CORPORATION (JP) 2009-12-30 WO disclosed