SCHEMBL1831228

SCHEMBL1831228

CC(C(=O)O)n1cnc2cncnc21

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
USP5 P45974 1/20 0.48
FDPS P14324 1/20 0.43
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
DNMT3B Q9UBC3 1/20 0.37
HCAR3 P49019 1/20 0.36
TSHR P16473 5/20 0.36
KDM4E B2RXH2 1/20 0.36
IRAK4 Q9NWZ3 1/20 0.35
CYP1A2 P05177 6/20 0.35
CYP3A4 P08684 6/20 0.35
CYP2C9 P11712 6/20 0.35
ALDH1A1 P00352 5/20 0.35
CYP2C19 P33261 4/20 0.35
LMNA P02545 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HBB P68871 1/20 0.35
CLK4 Q9HAZ1 2/20 0.34
HSD17B10 Q99714 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7457457 0.85 FDPS (0.42) USP5FDPSHDAC1HDAC6DNMT3B
SCHEMBL7455152 0.81 FDPS (0.42) USP5FDPSHDAC1HDAC6DNMT3B
SCHEMBL30539287 0.80 ADORA2A (0.47) FDPSHDAC1HDAC6HCAR3ALDH1A1
SCHEMBL754943 0.80 ADORA2A (0.47) FDPSHDAC1HDAC6HCAR3ALDH1A1
SCHEMBL5025564 0.77 FDPS (0.41) FDPSHDAC1HDAC6TSHRIRAK4
SCHEMBL7446654 0.76 FDPS (0.42) FDPSHDAC1HDAC6DNMT3BHCAR3
SCHEMBL28187328 0.75 FDPS (0.41) USP5FDPSHDAC1HDAC6DNMT3B
SCHEMBL7451329 0.75 FDPS (0.41) FDPSHDAC1HDAC6DNMT3BTSHR
SCHEMBL22571187 0.74 ADORA2A (0.53) FDPSHDAC1HDAC6TSHRKDM4E
SCHEMBL28038040 0.74 FDPS (0.43) FDPSHDAC1HDAC6DNMT3BTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2493895-A1 N-CONTAINING HETEROARYL DERIVATIVES AS JAK3 KINASE INHIBITORS Palau Pharma, S.A. (ES) 2012-09-05 EP disclosed
WO-2011051452-A1 N-CONTAINING HETEROARYL DERIVATIVES AS JAK3 KINASE INHIBITORS PALAU PHARMA, S.A. (ES) 2011-05-05 WO disclosed