SCHEMBL18315430

SCHEMBL18315430

CCC(c1ccccc1)n1nnc(C(=O)O)c1C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.50
TP53 P04637 1/20 0.44
ALOX12 P18054 1/20 0.44
KDM4C Q9H3R0 1/20 0.40
OPRM1 P35372 1/20 0.39
OPRD1 P41143 1/20 0.39
OPRK1 P41145 1/20 0.39
OPRL1 P41146 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ASPH Q12797 1/20 0.38
KDM8 Q8N371 1/20 0.38
HPGD P15428 1/20 0.38
HCAR3 P49019 2/20 0.37
ITK Q08881 2/20 0.37
ATM Q13315 2/20 0.37
CYP19A1 P11511 1/20 0.37
SLC5A1 P13866 1/20 0.37
SLC5A2 P31639 1/20 0.37
BRD4 O60885 2/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23130729 0.71 HTT (0.47) HTTTP53ALOX12HPGDHCAR3
SCHEMBL27858982 0.70 PTPN2 (0.52) ATM
SCHEMBL13027800 0.68 MEN1 (0.54) KDM4COPRM1OPRD1OPRK1OPRL1
SCHEMBL24460791 0.68 KLKB1 (0.45) TP53KDM4CKDM4EASPHKDM8
SCHEMBL4771303 0.67 HTT (1.00) HTTTP53ALOX12KDM4E
SCHEMBL24966874 0.67 TP53 (0.51) TP53ALOX12KDM4EHPGDCYP19A1
SCHEMBL24966930 0.67 TP53 (0.51) TP53ALOX12KDM4EHPGDCYP19A1
SCHEMBL23234141 0.67 TP53 (0.51) TP53ALOX12KDM4EHPGDCYP19A1
SCHEMBL795210 0.67 HPGD (0.68) HTTHPGDHCAR3CYP19A1
SCHEMBL3491684 0.67 ALDH1A1 (0.45) KDM4CKDM4EASPHKDM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2951185-B1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC (US) 2016-12-21 EP disclosed