SCHEMBL18323923

SCHEMBL18323923

CCC1CCC(NC(=O)c2ccncc2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.51
KDM4E B2RXH2 2/20 0.51
L3MBTL1 Q9Y468 1/20 0.50
ALDH1A1 P00352 1/20 0.49
GFER P55789 1/20 0.49
CYP46A1 Q9Y6A2 1/20 0.48
CYP19A1 P11511 1/20 0.48
NAMPT P43490 3/20 0.47
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC2 Q92769 1/20 0.47
NAAA Q02083 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46
GRM5 P41594 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1544549 0.87 L3MBTL1 (0.61) GAAKDM4EL3MBTL1ALDH1A1GFER
SCHEMBL621180 0.86 CYP46A1 (0.52) GAAKDM4EL3MBTL1ALDH1A1GFER
SCHEMBL25946525 0.85 GAA (0.49) GAAKDM4EL3MBTL1ALDH1A1GFER
SCHEMBL15014140 0.84 MEN1 (0.61) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL15014137 0.84 MEN1 (0.61) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL18387872 0.84 MEN1 (0.61) NPC1RAB9ASMN1; SMN2MEN1KMT2A
SCHEMBL23573442 0.84 CYP46A1 (0.56) GAAKDM4EL3MBTL1ALDH1A1GFER
SCHEMBL23573440 0.84 CYP46A1 (0.56) GAAKDM4EL3MBTL1ALDH1A1GFER
SCHEMBL12385843 0.83 GAA (0.55) GAAKDM4EL3MBTL1ALDH1A1GFER
SCHEMBL17133511 0.83 GAA (0.55) GAAKDM4EL3MBTL1ALDH1A1GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2922840-B1 BICYCLIC HETEROCYCLE SUBSTITUTED PYRIDYL COMPOUNDS USEFUL AS KINASE MODULATORS BRISTOL MYERS SQUIBB CO (US) 2016-12-21 EP disclosed