SCHEMBL18324497

SCHEMBL18324497

COC(=O)C(Cc1ccccn(S(=O)(=O)CC[SiH](C)C)ccc1)NC(=O)N1CCC(N2Cc3ccccc3NC2=O)CC1

nearest known ligand 0.52

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CALCA P06881 1/20 0.52
GAA P10253 1/20 0.49
CALCRL Q16602 17/20 0.48
CYP3A4 P08684 16/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18324498 0.84 CALCA (0.50) CALCACALCRLCYP3A4
SCHEMBL18324451 0.82 CALCA (0.49) CALCAGAACALCRLCYP3A4
SCHEMBL3282021 0.80 CALCA (0.60) CALCACALCRLCYP3A4
SCHEMBL3595749 0.78 CALCA (0.58) CALCACALCRLCYP3A4
SCHEMBL3607821 0.78 CALCRL (0.76) CALCACALCRLCYP3A4
SCHEMBL3607815 0.78 CALCRL (0.76) CALCACALCRLCYP3A4
SCHEMBL3587479 0.77 CALCRL (0.60) CALCACALCRLCYP3A4
SCHEMBL3591393 0.77 CALCA (0.57) CALCACALCRLCYP3A4
SCHEMBL3587476 0.77 CALCRL (0.60) CALCACALCRLCYP3A4
SCHEMBL3597734 0.77 CALCA (0.55) CALCAGAACALCRLCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539766-B1 CALCITONIN GENE RELATED PEPTIDE RECEPTOR ANTAGONISTS BRISTOL MYERS SQUIBB CO (US) 2016-12-21 EP disclosed