SCHEMBL1833797

SCHEMBL1833797

Nc1c[nH]c(-c2nc(NCC(c3ccccc3)c3ccccc3)c3ncn([C@@H]4C[C@H](NC(=O)CO)[C@@H](O)[C@H]4O)c3n2)n1

nearest known ligand 0.56

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.56
ADORA3 P0DMS8 10/20 0.56
ADORA1 P30542 4/20 0.44
ADORA2B P29275 3/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1830963 0.84 ADORA2A (0.65) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL241802 0.84 ADORA2A (0.65) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2883240 0.84 ADORA2A (0.60) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL241132 0.84 ADORA2A (0.60) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL240011 0.83 ADORA2A (0.57) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL293054 0.83 ADORA2A (0.55) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL1843512 0.82 ADORA2A (0.55) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL238863 0.82 ADORA2A (0.55) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL293561 0.81 ADORA2A (0.55) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL241166 0.81 ADORA2A (0.55) ADORA2AADORA3ADORA1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2322525-A1 Purine derivatives for use as adenosin A2A receptor agonists Novartis AG (CH) 2011-05-18 EP disclosed