SCHEMBL293561

SCHEMBL293561

Nc1cnn(-c2nc(NCC(c3ccccc3)c3ccccc3)c3ncn(C4CC(NC(=O)CO)C(O)C4O)c3n2)c1

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 16/20 0.55
ADORA3 P0DMS8 9/20 0.55
ADORA1 P30542 3/20 0.43
ADORA2B P29275 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL241166 1.00 ADORA2A (0.55) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL293560 1.00 ADORA2A (0.55) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL241667 0.94 ADORA2A (0.49) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL239220 0.94 ADORA2A (0.64) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL291925 0.91 ADORA2A (0.55) ADORA2AADORA3ADORA1
SCHEMBL2992492 0.90 ADORA2A (0.54) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL10158816 0.90 ADORA2A (0.54) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2992504 0.90 ADORA2A (0.54) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL2992497 0.90 ADORA2A (0.54) ADORA2AADORA3ADORA1ADORA2B
SCHEMBL292452 0.90 ADORA2A (0.55) ADORA2AADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2013211-B1 PURINE DERIVATIVES FOR USE AS ADENOSIN A2A RECEPTOR AGONISTS NOVARTIS AG (CH) 2012-03-14 EP disclosed