SCHEMBL18360682

SCHEMBL18360682

CCC1CC(C(=O)O)CN(Cc2c(F)cccc2F)C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 3/20 0.45
TSHR P16473 2/20 0.44
TDP1 Q9NUW8 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
S1PR1 P21453 10/20 0.44
S1PR5 Q9H228 6/20 0.44
S1PR3 Q99500 4/20 0.42
S1PR4 O95977 1/20 0.42
POLB P06746 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ALOX15 P16050 1/20 0.41
ENPP2 Q13822 1/20 0.41
GRK5 P34947 1/20 0.40
CDK8 P49336 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
EED O75530 1/20 0.40
PDE8A O60658 1/20 0.39
PDE8B O95263 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15084392 0.84 S1PR1 (0.46) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL10212863 0.83 S1PR5 (0.47) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL15081969 0.76 EED (0.39) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL15084388 0.75 CD274 (0.45) KDM4EL3MBTL1MEN1KMT2A
SCHEMBL2728895 0.74 CD274 (0.45) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL15084389 0.73 ALDH1A1 (0.46) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL15081966 0.71 ALDH1A1 (0.41) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL807578 0.71 ALDH1A1 (0.43) ALDH1A1KDM4ETSHRTDP1L3MBTL1
SCHEMBL15084390 0.70 EED (0.43) ALDH1A1KDM4ETSHRPOLBSMN1; SMN2
SCHEMBL807604 0.70 ALDH1A1 (0.50) ALDH1A1KDM4ETDP1L3MBTL1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2615916-B1 FUSED PYRAZOLE DERIVATIVES AS NOVEL ERK INHIBITORS MERCK SHARP & DOHME (US) 2017-01-04 EP disclosed