SCHEMBL18376830

SCHEMBL18376830

CS(=O)(=O)c1ccc(-c2cccc3cnc(Nc4ccc(OCCN5CCCC5)cc4)nc23)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
JAK2 O60674 11/20 0.68
JAK3 P52333 11/20 0.68
PTK2 Q05397 9/20 0.68
BRAF P15056 2/20 0.52
SRC P12931 4/20 0.52
BRD4 O60885 3/20 0.52
FGFR1 P11362 3/20 0.52
PDGFRB P09619 3/20 0.52
ABL1 P00519 3/20 0.52
EGFR P00533 3/20 0.52
YES1 P07947 3/20 0.52
KDR P35968 3/20 0.52
EPHB4 P54760 3/20 0.52
BRDT Q58F21 2/20 0.52
AXL P30530 2/20 0.52
MERTK Q12866 2/20 0.52
LCK P06239 2/20 0.52
FYN P06241 2/20 0.52
LYN P07948 2/20 0.52
RPS6KB1 P23443 2/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29371925 0.92 BRAF (0.60) JAK2JAK3PTK2BRAFSRC
SCHEMBL18377066 0.92 BRAF (0.60) JAK2JAK3PTK2BRAFSRC
SCHEMBL18376808 0.91 JAK2 (0.57) JAK2JAK3PTK2BRAFSRC
SCHEMBL18376653 0.91 JAK2 (0.57) JAK2JAK3PTK2BRAFSRC
SCHEMBL18377042 0.89 BRAF (0.55) JAK2JAK3PTK2BRAFSRC
SCHEMBL29370829 0.89 BRAF (0.55) JAK2JAK3PTK2BRAFSRC
SCHEMBL28679014 0.85 JAK2 (0.51) JAK2JAK3PTK2BRAFSRC
SCHEMBL18377069 0.85 JAK2 (0.57) JAK2JAK3PTK2BRAFSRC
SCHEMBL18376804 0.85 JAK2 (0.57) JAK2JAK3PTK2BRAFSRC
SCHEMBL18376823 0.85 SRC (0.53) JAK2JAK3PTK2BRAFSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017005137-A1 QUINAZOLINE COMPOUND, INTERMEDIATE, PREPARATION METHOD, PHARMACEUTICAL COMPOSITION AND USES THEREOF 吉林大学 2017-01-12 WO disclosed