SCHEMBL183845

SCHEMBL183845

COCCN(C(=O)O)[C@@H]1CCN(c2nc(-c3c(O)cccc3F)nc3cc(C)ccc23)C1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.58
JAK2 O60674 7/20 0.37
JAK3 P52333 6/20 0.37
FFAR4 Q5NUL3 1/20 0.33
HIF1A Q16665 1/20 0.33
JAK1 P23458 1/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
TP53 P04637 1/20 0.33
CTNNB1 P35222 2/20 0.32
TCF7L2 Q9NQB0 2/20 0.32
UBE2M P61081 1/20 0.32
DCUN1D1 Q96GG9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL183846 1.00 CHEK2 (0.58) CHEK2JAK2JAK3FFAR4HIF1A
SCHEMBL184160 0.89 CHEK2 (0.63) CHEK2JAK2JAK3MAPTUBE2M
SCHEMBL184161 0.89 CHEK2 (0.63) CHEK2JAK2JAK3MAPTUBE2M
SCHEMBL1622069 0.87 CHEK2 (0.51) CHEK2JAK2JAK3FFAR4KDM4E
SCHEMBL2733679 0.86 CHEK2 (0.57) CHEK2JAK2JAK3KDM4EMAPT
SCHEMBL5506872 0.86 CHEK2 (0.68) CHEK2JAK2JAK3MAPTMEN1
SCHEMBL4015698 0.86 CHEK2 (0.68) CHEK2JAK2JAK3MAPTMEN1
SCHEMBL1624102 0.84 CHEK2 (0.48) CHEK2KDM4EMAPTMEN1ALDH1A1
SCHEMBL1623249 0.84 CHEK2 (0.62) CHEK2JAK2JAK3HIF1AMAPT
Hydrochloric Acid SCHEMBL1624150 0.83 CHEK2 (0.47) CHEK2KDM4EMAPTMEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957482-B1 QUINAZOLINES USEFUL AS MODULATORS OF VOLTAGE GATED ION CHANNELS VERTEX PHARMA (US) 2012-01-04 EP disclosed