SCHEMBL184161

SCHEMBL184161

Cc1ccc2c(N3CCC(N(Cc4ccccc4)C(=O)O)C3)nc(-c3c(O)cccc3F)nc2c1

nearest known ligand 0.63

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 4/20 0.63
UBE2M P61081 8/20 0.39
DCUN1D1 Q96GG9 8/20 0.39
JAK2 O60674 1/20 0.38
JAK3 P52333 1/20 0.38
CCR5 P51681 4/20 0.37
KCNH2 Q12809 1/20 0.37
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL184160 1.00 CHEK2 (0.63) CHEK2UBE2MDCUN1D1JAK2JAK3
SCHEMBL183846 0.89 CHEK2 (0.58) CHEK2UBE2MDCUN1D1JAK2JAK3
SCHEMBL183845 0.89 CHEK2 (0.58) CHEK2UBE2MDCUN1D1JAK2JAK3
SCHEMBL5506872 0.88 CHEK2 (0.68) CHEK2JAK2JAK3MAPT
SCHEMBL4015698 0.88 CHEK2 (0.68) CHEK2JAK2JAK3MAPT
SCHEMBL1621663 0.88 CHEK2 (0.60) CHEK2CCR5KCNH2MAPT
Hydrochloric Acid SCHEMBL1624310 0.87 CHEK2 (0.59) CHEK2CCR5KCNH2MAPT
SCHEMBL1623249 0.86 CHEK2 (0.62) CHEK2JAK2JAK3MAPT
SCHEMBL1622398 0.83 CHEK2 (0.56) CHEK2MAPT
SCHEMBL4021314 0.83 CHEK2 (0.56) CHEK2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957482-B1 QUINAZOLINES USEFUL AS MODULATORS OF VOLTAGE GATED ION CHANNELS VERTEX PHARMA (US) 2012-01-04 EP disclosed