SCHEMBL18389

SCHEMBL18389

Nc1ccc(S(=O)(=O)N2CCN(c3ncc(C(O)(C(F)(F)F)C(F)(F)F)cn3)[C@@H](CN3C4COC[C@@H]3CC(O)C4)C2)s1

nearest known ligand 0.46

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
GCK P35557 9/20 0.46
GCKR Q14397 11/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12093442 1.00 GCK (0.46) GCKGCKR
SCHEMBL18415 1.00 GCK (0.46) GCKGCKR
SCHEMBL12093436 0.91 GCK (0.46) GCKGCKR
SCHEMBL16681 0.91 GCK (0.46) GCKGCKR
SCHEMBL12089546 0.91 GCK (0.46) GCKGCKR
SCHEMBL12089842 0.91 GCK (0.46) GCKGCKR
SCHEMBL18158 0.89 GCK (0.46) GCKGCKR
SCHEMBL12093446 0.89 GCK (0.46) GCKGCKR
SCHEMBL33228 0.89 GCK (0.46) GCKGCKR
SCHEMBL16804 0.86 GCKR (0.59) GCKGCKR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027261-A1 SULFONYLPIPERAZINE DERIVATIVES THAT INTERACT WITH GLUCOKINASE REGULATORY PROTEIN FOR THE TREATMENT OF DIABETES AMGEN INC. (US) 2012-03-01 WO disclosed